Symbol: |
GRK1
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Description: |
G protein-coupled receptor kinase 1 [Source:HGNC Symbol;Acc:10013]
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Location: |
Chr13:114321594-114438637[+]
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CRmiRSNP:
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Records:null
Compound |
CRmiRSNP |
SNP_sig |
Model |
Molecule |
Mol_sig |
Type |
Model : M1-Allele, M2-Recessive, M3-Additive, M4-Dominant
Total:0 Current:1
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Compound:
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Records:386
Gene |
Compound |
Gen_sig |
Exp_pattern |
GRK1 |
Dasatinib |
0.025 |
Up |
GRK1 |
NSC 732719 |
0.001 |
Down |
GRK1 |
NSC 733155 |
0.018 |
Down |
GRK1 |
gamma-glutamyl-alpha-amino-beta-[[2-ethyl(5-fluoro-2'deoxyur idyl) N-methyl-N-(4-chlorobutyl)phosphoramidoyl]sulfonyl] propionyl-(R)-(-)-phenylglycine |
0.001 |
Down |
GRK1 |
6-(3-Azido-propyl)-2,3-dimethoxthy-5,11-dioxo-5,11-dihydro-6 H-indeno[1,2-c]isoquinoline-9-carbonitrile |
0.033 |
Up |
GRK1 |
6-(3-Bromopropyl)-5,6-dihydro-9-methyl-3-nitro-5,11-dioxo-11 H-indeno[1,2-c]isoquinoline |
0.002 |
Down |
GRK1 |
4-[(Z)-2-(5-nitro-2-furyl)ethenyl]-6-(4-phenylpiperazin-1-yl )-1,3,5-triazin-2-ylamine |
0.027 |
Down |
GRK1 |
6-(3-Aminopropyl)-5,6-dihyro-9-iodo-3-nitro-5,11-dioxo-11H-i ndeno[1,2-c]isoquinoline Hydrochloride |
0.031 |
Down |
GRK1 |
6-(3-Aminopropyl)-5,6-dihydro-3-nitro-5,11-dioxo-9-thiomethy l-11H-indeno[1,2-c]isoquinoline Hydrochloride |
0.004 |
Down |
GRK1 |
7-(2-Pyrrolidinoethyl)oximino-5-androsten-3b,17b-diol diacetate |
0.023 |
Down |
GRK1 |
6-(3-Chloropropyl)-5,6-dihydro-2,3,9-trimethoxy-5,11-dioxo-1 1H-indeno[1,2-c]isoquinoline |
0.017 |
Down |
GRK1 |
6-[3-[2-[1,2,4]-Triazolyl-1-propyl]-5,6-dihydro-2,3-dimethox y-8,9-methylenedioxy-5,11-dioxo-11H-indeno[1,2-c]isoquinolin e Hydrochloride |
0.028 |
Down |
GRK1 |
6-(3-Aminopropyl)-5,6-dihbydro-3-nitro-5,11-dioxo-9-phenyl-1 1H[1,2-c]isoquinoline Hydrochloride |
0.001 |
Down |
GRK1 |
6-(10'-tert-BOC-aminododecyl)-5,6-dihydro-5,11-dioxo-11H-indeno-[1,2-c]isoquinoline |
0.046 |
Up |
GRK1 |
5,6-Dihydro-6-[3-(2-hydroxyethyl)amino-1-propyl]-3-nitro-5,11-dioxo-11H-indeno[1,2-c]isoquinoline Hydrochloride |
0.011 |
Down |
Expression pattern: Sensitivity / Resistance
Total:26 Current:24
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SNP:
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Records:null
SNP |
Gene |
SNP_location |
SNP_allele |
Total:0 Current:1
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miRNA:
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Records:6
Gene |
Gen_transcript |
miRNA |
miR_location |
GRK1 |
ENST00000335678 |
hsa-mir-512-5p |
Chr19:54169946-54169968[+] |
GRK1 |
ENST00000335678 |
hsa-mir-512-5p |
Chr19:54172430-54172452[+] |
GRK1 |
ENST00000335678 |
hsa-mir-566 |
Chr3:50210774-50210792[+] |
GRK1 |
ENST00000335678 |
hsa-mir-615-3p |
Chr12:54427794-54427815[+] |
GRK1 |
ENST00000335678 |
hsa-mir-941 |
Chr20:62550848-62550870[+] |
GRK1 |
ENST00000335678 |
hsa-mir-941 |
Chr20:62551155-62551177[+] |
Total:1 Current:1
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